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Ionizable networks mediate pH-dependent allostery in the SH2 domain-containing signaling proteins SHP2 and SRC.

Van Dyck PK, Piszkin L, Gorski EA, Nascimento ET, Abebe JA, Hoffmann LM, Peng JW, White KA
Sci Signal. 2025 Nov 11;18(912):eadt3018. doi: 10.1126/scisignal.adt3018. Epub 2025 Nov 11. (Link opens in a new window) PubMed (Link opens in a new window) Article

Plasmids from Article

ID Plasmid Purpose
244491pGEX-4T1 SHP2 E252ABacterial Expression of SHP2 mutant
244492pGEX-4T1 GST-SHP2 H116ABacterial Expression of SHP2 mutant
244493pGEX-4T1 GST-SHP2 H116A E252ABacterial Expression of pH insensitive SHP2 mutant
246423Flag-Src C185AExpresses Src mutant C185A or C188A in Mammalian cells
246424Flag-Src H201AExpresses Src mutant H201A (aka H204A) in Mammalian cells
246425Flag- Src H492AExpresses Src mutant H492A (aka H495A) in Mammalian cells
246426Flag-Src E524AExpresses Src mutant E524A (aka E527A) in Mammalian cells
246427Flag-Src C185A H201A H492A E524AExpresses Src pH insensitive mutant in Mammalian cells
246428Flag-Src Y527EExpresses Src mutant Y527E (aka Y530E) in Mammalian cells
246429Flag-Src Y527AExpresses Src mutant Y527A (aka Y530A) in Mammalian cells

Antibodies from Article