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Manipulation of very few receptor discriminator residues greatly enhances receptor specificity of non-visual arrestins.

Gimenez LE, Vishnivetskiy SA, Baameur F, Gurevich VV
J Biol Chem. 2012 Aug 24;287(35):29495-505. doi: 10.1074/jbc.M112.366674. Epub 2012 Jul 11. (Link opens in a new window) PubMed (Link opens in a new window) Article

Plasmids from Article

ID Plasmid Purpose
234807p3HM2LucMammalian expression of human muscarinic M2 receptor fused to RLuc8
234808p3HB2ALucMammalian expression of human B2-adrenergic receptor fused to RLuc8
236275p3HAT1Luc1Mammalian expression of human angiotensin II type 1 receptor; N-terminal HA tag, C-terminal Rluc8
236276p3HD1RLuc2Mammalian expression of human dopamine D1 receptor; N-terminal HA tag, C-terminal Rluc8
236277p3HM1Luc4Mammalian expression of human muscarinic M1 receptor; N-terminal HA tag, C-terminal Rluc8

Antibodies from Article